Drug class: Aromatase Inhibitor Common names: Aromadex, Aromasin, Aromasine, Aromaxyl, Exemestane, Examestane Chemical structure: 6-methyleneandrosta-1,4-diene-3,17-dio …
Info: Exemestane is a steroidal Aromatase Inhibitor (AI) that is most commonly known as Aromasin.
Exemestane was first released on the U.S. market in 2000 after shortly gaining FDA approval a few months prior in 1999. The primary purpose of use as with most AI’s would be to combat breast cancer in post-menopausal women. Shortly after, the AI would begin to gain a lot of popularity among anabolic steroid users for its ability to protect against estrogenic related side effects.
This action is very similar to the older and more popular AI’s in Arimidex (Anastrozole). It would also gain a fair amount of popularity during Cycle and in Post Cycle Therapy (PCT) plans among steroid users. It was not the first AI to gain such popularity but would prove to be a little more advantageous for this purpose than most AI’s
- Androgenic index – low
- Anabolic index n/a
- Estrogen level – n/a (exemestane as an estrogen blocker)
- Progestogens activity – n/a
- Toxicity for the liver – low
Exemestane – a new generation of drug that blocks enzymes responsible for aromatisation.
As a result of the drug are suppressed 80-85% estrogens in the body of the athlete.
DOSE RANGE AND DURATION OF USE
It is recommended to take Exemestan during meals or after meal.
Common cycle length is 2-4 weeks (some getting only two to three doses per week)
Beginners: 12.5mg / EOD (every other day)
Hobby: 12.5 mg / ED (every day)
Professional Range: 25 mg / ED (every day)
Women: 12.5mg / ED or EOD
Half-life: 25-27 hours (active life about 130 hours)
Detection time: 2-3 weeks
Weakness or Fatigue
High Blood Pressure
Nausea and/or Vomiting (rare)
AFTER CYCLE THERAPY
Exemestane can be part of your cycle. (Exemestane during steroid cycle prevents the side effects that steroids can cause – flavoring).
Also Exemestane can be used as Post Cycle Therapy.
To be store in a dry place, protected from light, at a temperature of 15-25 ° C. Keep out of reach of children.
MIX/COMBINE YOUR STEROIDS CYCLE
Exemestan use is not limited to PCT only, it also can be a part of your steroid cycle. It outperform Arimidex with about 12 % when it comes to estrogen inhibition. And it will even cause an increase of testosterone level as well. But Exemestan is a steroidal drug, which mean it carry on androgenic effects too. That’s why the best will be to let ti for PCT time, when this trait would be even beneficial.